KT5823

货号： 2164-250      产品名称： KT5823   品牌： Biovision 规格： 250 μg 3周到货 生化实验

KT5823
A protein kinase G (PKG) inhibitor
Product Overview
Product Name: KT5823
Alternate Name/Synonyms: 2,​3,​9,​10,​11,​12-​hexahydro-​10R-​methoxy-​2,​9-​dimethyl-​1-​oxo-​ 9S,​12R-​epoxy-​1H-​diindolo[1,​2,​3-​fg:3’,​2’,​1’-​kl]pyrrolo[3,​4-​ i][1,​]benzodiazocine-​10-​carboxylic acid,​ methyl ester
Description: Cell-permeable. KT5823 is a derivative of K-252a (Cat. No. 2013) that acts as a selective inhibitor of Protein kinase G (PKG) (Ki = 0.234 µM). Inhibits other kinases at much higher concentrations (Ki’s for PKA = 4 μM and for MLCK=>10 μM).
Peptide Sequence: N/A
Appearance: White solid
Formulation: N/A
CAS Number: 126643-37-6
Molecular Formula: C₂₉H₂₅N₃O₅
Molecular Weight: 495.53
Purity: ≥98% by HPLC
Solubility:DMSO (20 mg/ml)
Storage Temp.: -20°C
Shipping Conditions: gel pack
Handling: Protect from air and light
SMILES: CC12C(CC(O1)N3C4=CC=CC=C4C5=C6C(=C7C8=CC=CC=C8N2C7=C53)CN(C6=O)C)(C(=O)OC)OC
InChi: InChI=1S/C29H25N3O5/c1-28-29(36-4,27(34)35-3)13-20(37-28)31-18-11-7-5-9-15(18)22-23-17(14-30(2)26(23)33)21-16-10-6-8-12-19(16)32(28)25(21)24(22)31/h5-12,20H,13-14H2,1-4H3
InChi Key: QTYMDECKVKSGSM-UHFFFAOYSA-N
PubChem CID: 3843
MDL Number: MFCD09878278
USAGE: For Research Use Only! Not For Use in Humans.

-20°C